| ANTICONVULSANT AGENTS |
| Carbamazepine (Equetro®, Tegretol®) | Off-label use | | | Off-label use | |
| Divalproex sodium (Depakote®) | Off-label use | | | Off-label use | |
| Gabapentin (Neurontin®) | Off-label use | | | | Off-label use |
| Pregabalin (Lyrica®) | Off-label use | | | | |
| Tiagabine (Gabitril®) | Off-label use | | | | |
| ANTIDEPRESSANT AGENTS |
| Amitriptyline (Elavil®) | Off-label use | | Off-label use | Off-label use | |
| Amoxapine (Asendin®) | Off-label use | | Off-label use | Off-label use | |
| Citalopram (Celexa®) | Off-label use | Off-label use | Off-label use | Off-label use | Off-label use |
| Clomipramine HCl (Anafranil®) | Off-label use | FDA approved | Off-label use | Off-label use | Off-label use |
| Desipramine (Norpramin®, Pertofrane®) | Off-label use | | Off-label use | Off-label use | |
| Desvenlafaxine (Pristiq®) | Off-label use | Off-label use | Off-label use | Off-label use | Off-label use |
| Doxepin (Adapin ®, Sinequan®) | Off-label use | | Off-label use | Off-label use | Off-label use |
| Duloxetine HCl (Cymbalta®) | FDA approved | Off-label use | Off-label use | Off-label use | Off-label use |
| Escitalopram oxalate (Lexapro®) | FDA approved | Off-label use | Off-label use | Off-label use | Off-label use |
| Fluoxetine HCl (Prozac®, Prozac® Weekly™) | Off-label use | FDA approved | FDA approved | Off-label use | Off-label use |
| Fluvoxamine (Luvox®, Luvox CR®) | Off-label use | FDA approved | Off-label use | Off-label use | FDA approved |
| Imipramine (Tofranil®) | Off-label use | | Off-label use | Off-label use | Off-label use |
| Isocarboxazid (Marplan®) | | | Off-label use | | Off-label use |
| Maprotiline HCl (Ludiomil®)a | Off-label use | | Off-label use | Off-label use | |
| Milnacipran (Savella®) | Off-label use | Off-label use | Off-label use | Off-label use | Off-label use |
| Mirtazapine (Remeron®, Remeron SolTab®) | Off-label use | Off-label use | Off-label use | Off-label use | |
| Nefazodone (Serzone®) | Off-label use | | Off-label use | Off-label use | |
| Nortriptyline (Aventyl®, Pamelor®) | Off-label use | | Off-label use | Off-label use | |
| Paroxetine HCl (Paxil®, Paxil CR®) | FDA approved | FDA approved | FDA approved | FDA approved | FDA approved |
| Phenelzine (Nardil®) | Off-label use | | Off-label use | | Off-label use |
| Sertraline HCl (Zoloft®) | Off-label use | FDA approved | FDA approved | FDA approved | FDA approved |
| Tranylcypromine (Parnate®) | Off-label use | | Off-label use | | Off-label use |
| Trazodone (Desyrel®, Oleptro®) | Off-label use | | | | |
| Trimipramine (Surmontil®) | Off-label use | | Off-label use | | |
| Venlafaxine HCl (Effexor®, Effexor XR®) | FDA approved | Off-label use | FDA approved | Off-label use | FDA approved |
| Vilazodone (Viibryd®) | Off-label use | | | | |
| ANTIPSYCHOTIC AGENTS |
| Chlorpromazine (Thorazine®) | Off-label use | | | Off-label use | |
| Fluphenazine (Prolixin®) | | Off-label use | | Off-label use | |
| Haloperidol (Haldol®) | | Off-label use | | Off-label use | |
| Olanzapine (Zyprexa®) | Off-label use | Off-label use | | Off-label use | |
| Quetiapine (Seroquel®, Seroquel XR®) | Off-label use | | | Off-label use | |
| Risperidone (Risperdal®, Risperdal® Consta®) | | Off-label use | | Off-label use | |
| Trifluoperazine (Stelazine®) | FDA approved | | | Off-label use | |
| BENZODIAZEPINES |
| Alprazolam (Alprazolam Intensol®, Xanax®) | FDA approved | | FDA approved | | Off-label use |
| Clonazepam (Klonopin®)b | Off-label use | | FDA approved | | Off-label use |
| Clorazepate (Tranxene®) | FDA approved | | Off-label use | | Off-label use |
| Diazepam (Diazepam Intensol®, Valium®)b | FDA approved | | Off-label use | | Off-label use |
| Halazepam (Paxipam®) | FDA approved | | | | |
| Lorazepam (Ativan®, Lorazepam Intensol®) | FDA approved | | Off-label use | | Off-label use |
| Oxazepam (Serax ®)b | FDA approved | | Off-label use | | Off-label use |
| NONBENZODIAZEPINES |
| Buspirone HCl (BuSpar®, BuSpar® Dividose) | FDA approved | Off-label use | Off-label use | | Off-label use |
| Chlordiazepoxide (Librax®, Librium®, Limbitrol®, Limbitrol® DS)b | FDA approved | | Off-label use | | Off-label use |
| Diphenhydramine (Benadryl®) | Off-label use | | | | |
| Hydroxyzine (Anx®, Atarax®, Atarax® Syrup, Vistaril®)b, c | Off-label use | | | | |
| Meprobamate (Miltown ®) | FDA approved | | | | |
| Propranolol (Inderal ®) | Off-label use | | Off-label use | Off-label use | Off-label use |